TG4-155 62175 ClH/c1-3-19-15-24-22(23(4-2)27-19)13-14-25(33)32(24)16-17-9-11-18(12-10-17)20-7-5-6-8-21(20)26-28-30-31-29-26

ClH/c1-3-19-15-24-22(23(4-2)27-19)13-14-25(33)32(24)16-17-9-11-18(12-10-17)20-7-5-6-8-21(20)26-28-30-31-29-26

Chemical Name: (2R)-2-[(1H-1

Solubility: DMSO : 2 mg/mL (9

Methoprene elicits significant toxicity to endocrine-related processes in the 5-50 nM concentration range

23)24/h9-12

TG4-155 62175 ClH/c1-3-19-15-24-22(23(4-2)27-19)13-14-25(33)32(24)16-17-9-11-18(12-10-17)20-7-5-6-8-21(20)26-28-30-31-29-26TG4 155 is a potent, brain permeant and selective EP2 receptor antagonist with a Ki of 9. 9 nM. TG4 155 shows low nanomolar antagonist activity against only EP2 and DP1. TG4 155 has an EP2 Schild KB of 2. 4 nM and displays 550 4750 fold selectivity for EP2 over EP1, EP3, EP4 and IP, but only 14 fold selectivity against the DP1 receptor. Product information CAS Number: 1164462 05 8 Molecular Weight: 394. 46 Formula: C23H26N2O4 Chemical Name: (2E) N [2