DREADD agonist 21 has excellent bioavailability
Chemical Name: 2-(2-methoxy-4-{[(5E)-4-oxo-2-sulfanylidene-1
Smiles: O=C(C1C=CC(F)=CC=1)N1CC2OC(COC3C=CC=CC=3)=NC=2CC1
Chemical Name: 4-(4-{3-[2-(2
Halofuginone (0
INT-777 R-enantiomer clocycline Hydrochloride DREADD agonist 21 has excellentINT 777 (R enantiomer) is the R enantiomer of INT 777, with EC50 of 4. 79 M for TGR5, and less potent than INT 777. Product information CAS Number: 1198786 98 9 Molecular Weight: 450. 65 Formula: C27H46O5 Chemical Name: (2R,4R) 4 [(1R,3aS,3bR,4R,5R,5aS,7R,9aS,9bS,11S,11aR) 5 ethyl 4,7,11 trihydroxy 9a,11a dimethyl hexadecahydro 1H cyclopenta[a]phenanthren 1 yl] 2 methylpentanoic acid Smiles: